Synthesis of Phosphoisosteres of Amyloid Dipeptide Components

Мұқаба

Дәйексөз келтіру

Толық мәтін

Ашық рұқсат Ашық рұқсат
Рұқсат жабық Рұқсат берілді
Рұқсат жабық Рұқсат ақылы немесе тек жазылушылар үшін

Аннотация

A simple and effective method was proposed for the synthesis of new phosphinic peptides in free form, structural isosteres of the dipeptide components of beta-amyloid (Aβ42), potential inhibitors of zinc-metalloproteinases.

Толық мәтін

Рұқсат жабық

Авторлар туралы

S. Golovash

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
Ресей, Chernogolovka

D. Ivanov

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
Ресей, Chernogolovka

A. Borodachev

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
ORCID iD: 0000-0002-3458-5129
Ресей, Chernogolovka

V. Shestov

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
Ресей, Chernogolovka

M. Dmitriev

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
ORCID iD: 0000-0001-8870-195X
Ресей, Chernogolovka

V. Ragulin

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Хат алмасуға жауапты Автор.
Email: rvalery@dio.ru
ORCID iD: 0000-0002-3967-1034
Ресей, Chernogolovka

Әдебиет тізімі

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